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Category: EnzymesarrowKinasesarrowMyosin Light Chain Kinase
Cat.No. Product Name
1885 MLCK inhibitor peptide 18
Alternative name(s): Myosin Light Chain Kinase Inhibitor Peptide 18
Price and Availability

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MLCK Inhibitor Peptide 18

Biological Activity:

Selective competitive inhibitor of myosin light chain kinase (IC50 = 50 nM). Displays 4000-fold selectivity over CaM kinase II and does not inhibit PKA.

Technical Data:

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M.Wt: 1324.64
Formula: C60H105N23O11
Storage: Desiccate at -20°C
CAS No: [224579-74-2]

Resources:

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    • Certificate of Analysis / MSDS:

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    References:

    Lukas et al (1999) Identification of novel classes of protein kinase inhibitors using combinatorial peptide chemistry based on functional genomics knowledge. J.Med.Chem. 42 910.
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    Keywords: MLCK Inhibitor Peptide 18, Kinases, Selective Inhibitor Of Myosin Light Chain Kinase, Myosin Light Chain Kinase Inhibitor Peptide 18, Tocris Bioscience
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