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Category: Ion ChannelsarrowLigand-gated Ion ChannelsarrowGlutamate (Ionotropic) ReceptorsarrowNMDA SelectivearrowNMDA SitearrowAntagonists
Cat.No. Product Name
1019 LY 235959
Price and Availability

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LY 235959

Other Information:

Sold with the permission of Eli Lilly and Company
Chemical Name: [3S-(3a,4aa,6b,8aa)]-Decahydro-6-(phosphonomethyl)-3-is oquinolinecarboxylic acid)

Biological Activity:

Competitive NMDA receptor antagonist.

Technical Data:

 Click here for more information on batch specific data
M.Wt: 277.26
Formula: C11H20NO5P
Storage: Desiccate at +4°C
Solubility: Soluble to 100 mM in Water
CAS No: [137433-06-8]

Resources:

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    • Certificate of Analysis / MSDS:

    Certificate of Analysis: View current batch
    Product/Material Safety Data Sheet: View current batch

    References:

    Ellison (1994) Competitive and non-competitive NMDA antagonists induce similar limbic degeneration. Neuroreport 5 2688. Borowicz et al (1996) Competitive NMDA-receptor antagonists, LY 235959 and LY 233053, enhance the protective efficacy of various antiepileptic drugs against maximal electroshock-induced seizures in mice. Epilepsia 37 618.

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    Keywords: LY 235959, Ligand-gated Ion Channels, Competitive NMDA Antagonist, LY235959, Tocris Bioscience
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