Click here for full price details of (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
Chemical Name:N-[(1R)-2-[[[(1S*,3R*)-3-(Aminomethyl)cyclohexyl]methyl
]amino]-1-(1H-indol-3-ylmethyl)-2-oxoethyl]spiro[1H-ind
ene-1,4'-piperidine]-1'-carboxamide
Biological Activity:
Potent and selective somatostatin sst2
receptor agonist (Ki values are 4, 537, 2480, 3614 and 5017 nM for
cloned human sst2, sst1, sst4, sst3
and sst5 receptors respectively).
Yanget al
(1998) Spiro[1H-indene-1,4'-piperidine] derivatives as potent and
selective non-peptide human somatostatin receptor subtype 2 (sst2)
agonists. J.Med.Chem. 41 2175.
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