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Category: 7TM Receptorsarrow5-HT Receptorsarrow5-HT1 Receptorsarrow5-HT1A
Cat.No. Product Name
0797 8-Hydroxy-PIPAT oxalate  
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8-Hydroxy-PIPAT

Other Information:

Sold with the permission of the University of Pennsylvania
Chemical Name: (RS)-trans-8-Hydroxy-2-[N-n-propyl-N-(3'-iodo-2'-propen yl)amino]tetralin oxalate

Biological Activity:

High affinity 5-HT1A receptor agonist (Kd = 0.38 nM).

Technical Data:

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M.Wt: 461.3
Formula: C16H22INO.C2H2O4
Storage: Desiccate at -20°C
Solubility: Soluble to 100 mM in Ethanol and to 100 mM in DMSO
Purity: >98%
CAS No: [159651-91-9]

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    • Certificate of Analysis / MSDS:

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    References:

    Zhuang et al (1993) Synthesis of (R,S)-trans-8-Hydroxy-2-[N-n-propyl-N-(3'-iodo-2'-propenyl)amino]tetralin (trans-8-OH-PIPAT): a new 5-HT1A receptor ligand. J.Med.Chem. 36 3161.
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    Keywords: 8-Hydroxy-PIPAT, 5-HT Receptors, High Affinity 5-HT1A Agonist, 8Hydroxy-PIPAT, Tocris Bioscience
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