7-Hydroxy-PIPAT Maleate | Dopamine Receptors | D3 Agonist (D3 > D2) | 7-OH-PIPAT | 7Hydroxy-PIPAT Maleate

Category:

7TM Receptors

Dopamine Receptors

D2-like Receptors

D3-selective

Cat.No.

Product Name

0719

7-Hydroxy-PIPAT maleate

Alternative name(s):

7-OH-PIPAT

7-Hydroxy-PIPAT maleate
C16H22INO.C4H4O4 (RS)-trans-7-Hydroxy-2-[N-propyl-N-(3'-iodo-2'-propenyl)amino]tetralin maleate

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7-Hydroxy-PIPAT maleate

Other Information:

Sold with the permission of the University of Pennsylvania

Chemical Name: (RS)-trans-7-Hydroxy-2-[N-propyl-N-(3'-iodo-2'-propenyl )amino]tetralin maleate

Biological Activity:

This ligand has uniquely high affinity and selectivity for the D₃ receptor.

Technical Data:

M.Wt:	487.33
Formula:	C₁₆H₂₂INO.C₄H₄O₄
Storage:	Desiccate at +4°C
Solubility:	Soluble in DMSO
CAS No:	[159559-71-4]

Resources:

Certificate of Analysis / MSDS:

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References:

Foulon et al (1993) Synthesis of (R,S)-2'-trans-7-hydroxy-[N-(3'-iodo-2'-propenyl)-N-n-propyl]aminotetralin (trans-7-OH-PIPAT). J.Med.Chem. 36 1499. Chumpradit et al (1993) Synthesis and optical resolution of (R)- and (S)-trans-7-hydroxy-2-[N-propyl-N-(3'-iodo-2'-propenyl)amino]tetralin: a new D₃ dopamine receptor ligand. J.Med.Chem. 36 4308. Kung et al (1993) In vitro binding of a novel dopamine D₃ receptor ligand: [¹²⁵I]-trans-7-OH-PIPAT. Eur.J.Pharmacol. 235 165.

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Keywords: 7-Hydroxy-PIPAT Maleate, Dopamine Receptors, D3 Agonist (D3 > D2) , 7-OH-PIPAT, 7Hydroxy-PIPAT Maleate, Tocris Bioscience

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