Endomorphin-2 | Opioid Receptors | Potent & Selective M Agonist

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Cat.No.	Product Name
1056	Endomorphin-2

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Endomorphin-2

Biological Activity:

Endogenous peptide with extremely high affinity and selectivity for μ-opioid receptors (with K_i values of 0.69, 9233 and 5240 nM for μ, δ and κ respectively).

Technical Data:

M.Wt:	571.65
Formula:	C₃₂H₃₇N₅O₅
Storage:	Desiccate at -20°C
CAS No:	[141801-26-5]

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Certificate of Analysis / MSDS:

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References:

Zadina et al (1997) A potent and selective endogenous agonist for the µ-opiate receptor. Nature 386 499. Zadina et al (1997) A potent and selective endogenous agonist for the µ-opiate receptor. Nature 386 499. Chapman et al (1997) Distinct inhibitory effects of spinal endomorphin-1 and endomorphin-2 on evoked dorsal horn neuronal responses in the rat. Br.J.Pharmacol. 122 1537. Goldberg et al (1998) Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J.Pharmacol.Exp.Ther. 286 1007.

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Keywords: Endomorphin-2, Opioid Receptors, Potent & Selective M Agonist, Tocris Bioscience

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Opioid Receptors
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