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Category: Ion ChannelsarrowLigand-gated Ion ChannelsarrowGABAA and GABAC ReceptorsarrowBenzodiazepines
Cat.No. Product Name
2805 Diazepam
Alternative name(s): Ro 5-2807
Price and Availability

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Diazepam

Other Information:

This is a controlled substance in some countries with associated conditions of supply; the relevent licence/documentation from the appropriate governing body will be required.
Chemical Name: 7-Chloro-1-methyl-5-phenyl-3H-1,4-benzodiazepin-2(1H)-o ne

Biological Activity:

Ligand at the GABAA receptor benzodiazepine modulatory site. Anxiolytic, anticonvulsant and sedative/hypnotic agent.

Technical Data:

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M.Wt: 284.74
Formula: C16H13ClN2O
Storage: Store at RT
Solubility: Soluble to 100 mM in DMSO and to 25 mM in Ethanol
Purity: >98%
CAS No: [439-14-5]

Resources:

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    • Certificate of Analysis / MSDS:

    Certificate of Analysis is currently unavailable on-line. Please contact Customer Service
    Product/Material Safety Data Sheet: View current batch

    References:

    Sieghart et al (1994) Pharmacology of benzodiazepine receptors: an update. J.Psychiat.Neurosci. 19 24.
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    Keywords: Diazepam, Ligand-gated Ion Channels, Benzodiazepine Agonist, Ro 5-2807, Tocris Bioscience
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