Cyproheptadine Hydrochloride | 5-HT Receptors | 5-HT2 Antagonist

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Cat.No.	Product Name
0996	Cyproheptadine hydrochloride

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Cyproheptadine hydrochloride

Chemical Name: 4-(5H-Dibenzo[a,d]cyclohepten-5-ylidine)-methylpiperid ine hydrochloride

Biological Activity:

Non-selective 5HT₂ antagonist, migraine prophylactic.

Technical Data:

M.Wt:	323.86
Formula:	C₂₁H₂₁N.HCl
Storage:	Store at RT
Solubility:	Soluble to 15 mM in Water
Purity:	>98%
CAS No:	[969-33-5]

Resources:

Certificate of Analysis / MSDS:

Certificate of Analysis: View current batch

Product/Material Safety Data Sheet: View current batch

References:

Merck Index 12 2842. Hoyer et al (1994) VII. International Union of Pharmacology classification of receptors for 5-hydroxytryptamine (serotonin). Pharmacol.Rev. 46 157. Moran et al (1994) Inhibitory 5-hydroxytryptamine receptors involved in pressor effects obtained by stimulation of sympathetic outflow from spinal cord in pithed rats. Br.J.Pharmacol. 113 1358.

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Keywords: Cyproheptadine Hydrochloride, 5-HT Receptors, 5-HT2 Antagonist, Tocris Bioscience

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5-HT Receptors & their Ligands
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