Cinanserin Hydrochloride | 5-HT Receptors | Selective 5-HT2 Antagonist

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Cat.No.	Product Name
0460	Cinanserin hydrochloride

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Cinanserin hydrochloride

Chemical Name: N-[2-[[3-(Dimethylamino)propyl]thio]phenyl]-3-phenyl-2- propenamide hydrochloride

Biological Activity:

5-HT₂ antagonist.

Technical Data:

M.Wt:	376.94
Formula:	C₂₀H₂₄N₂OS.HCl
Storage:	Desiccate at RT
Solubility:	Soluble to 50 mM in Water
Purity:	>99%
CAS No:	[1166-34-3]

Resources:

Certificate of Analysis / MSDS:

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Product/Material Safety Data Sheet: View current batch

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References:

Leysen et al (1981) Receptor binding profile of R-41-468, a novel antagonist at 5HT₂ receptors. Life Sci. 28 1015. Pierce et al (1992) Molecular structure basis of ligand selectivity for 5-HT₂ versus 5-HT_1C cortical receptors. Naunyn-Schmied.Arch.Pharmacol. 346 4.

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Keywords: Cinanserin Hydrochloride, 5-HT Receptors, Selective 5-HT2 Antagonist, Tocris Bioscience

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5-HT Receptors & their Ligands
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