Carbetapentane Citrate | Sigma & Imidazoline | High Affinity S1 Ligand | Pentoxyverine Citrate

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Sigma and Imidazoline

Sigma Ligands

Sigma1

Cat.No.

Product Name

0454

Carbetapentane citrate

Alternative name(s):

Pentoxyverine citrate

Carbetapentane citrate
C20H31NO3.C6H8O7 1-Phenylcyclopentanecarboxylic acid 2-(2-diethylaminoethoxy)ethyl ester citrate

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Carbetapentane citrate

Chemical Name: 1-Phenylcyclopentanecarboxylic acid 2-(2-diethylaminoethoxy)ethyl ester citrate

Biological Activity:

A selective ligand for the σ₁-site.

Technical Data:

M.Wt:	525.59
Formula:	C₂₀H₃₁NO₃.C₆H₈O₇
Storage:	Store at RT
Solubility:	Soluble to 75 mM in DMSO
Purity:	>99%
CAS No:	[23142-01-0]

Resources:

Certificate of Analysis / MSDS:

Certificate of Analysis: View current batch

Product/Material Safety Data Sheet: View current batch

References:

Rothman et al (1991) Labelling by [³H]1,3-di(2-tolyl)guanidine of two high affinity binding sites in guinea pig brain: evidence for allosteric regulation by calcium channel antagonists and pseudoallosteric modulation by σ ligands. Mol.Pharmacol. 39 222. Quirion et al (1992) A proposal for the classification of sigma binding sites. TiPS 13 85.

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Keywords: Carbetapentane Citrate, Sigma & Imidazoline, High Affinity S1 Ligand, Pentoxyverine Citrate, Tocris Bioscience

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