CYN 154806 | Peptides (Hypothalamic / Pituitary Hormones) | Selective Sst2 Antagonist | CYN154806

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Category:

7TM Receptors

Peptides (Hypothalamic/Pituitary Hormones)

Somatostatin Receptors

Cat.No.	Product Name
1843	CYN 154806

Price and Availability

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CYN 154806

Biological Activity:

Potent and selective somatostatin sst₂ receptor antagonist. pIC₅₀ values are 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst₂, sst₁, sst₃, sst₄ and sst₅ receptors respectively.

Technical Data:

M.Wt:	1197.35
Formula:	C₅₆H₆₈N₁₂O₁₄S₂
Storage:	Desiccate at -20°C
CAS No:	[183658-72-2]

Resources:

Certificate of Analysis / MSDS:

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References:

Bass et al (1996) Identification and characterization of novel somatostatin antagonists. Mol.Pharmacol. 50 709. Feniuk et al (2000) Selective somatostatin sst₂ receptor blockade with the novel cyclic octapeptide, CYN-154806. Neuropharmacology 39 1443. Hannon et al (2002) Drug design at peptide receptors. Somatostatin receptor ligands. J.Mol.Neurosci. 18 15.

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Keywords: CYN 154806, Peptides (Hypothalamic / Pituitary Hormones), Selective Sst2 Antagonist, CYN154806, Tocris Bioscience

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Product Feature

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