CP 93129 Dihydrochloride | 5-HT Receptors | 5-HT1B Agonist | CP93129 Dihydrochloride

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Cat.No.	Product Name
1032	CP 93129 dihydrochloride

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CP 93129 dihydrochloride

Chemical Name: 1,4-Dihydro-3-(1,2,3,6-tetrahydro-4-pyridinyl)-5H-pyrro l[3,2-b]pyridin-5-one dihydrochloride

Biological Activity:

Potent and highly selective 5-HT_1B agonist.

Technical Data:

M.Wt:	288.18
Formula:	C₁₂H₁₃N₃O₂.2HCl
Storage:	Desiccate at RT
Solubility:	Soluble to 100 mM in Water
CAS No:	[127792-75-0]

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Certificate of Analysis / MSDS:

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References:

Iyer and Bradberry (1996) Serotonin-mediated increase in prefrontal cortex dopamine release: pharmacological characterisation. J.Pharmacol.Exp.Ther. 277 40. Trillat et al (1997) Regulation of serotonin release in the frontal cortex and ventral hippocampus of homozygous mice lacking 5-HT_1B receptors: in vivo microdialysis studies. J.Neurochem. 69 2019. Lee et al (1998) Infusion of the serotonin_1B (5-HT_1B) agonist CP-93,129 into the parabrachial nucleus potently and selectively reduces food intake in rats. Psychopharmacology 136 304.

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Keywords: CP 93129 Dihydrochloride, 5-HT Receptors, 5-HT1B Agonist, CP93129 Dihydrochloride, Tocris Bioscience

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