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Category: Ion ChannelsarrowLigand-gated Ion ChannelsarrowGlutamate (Ionotropic) ReceptorsarrowNMDA SelectivearrowNMDA SitearrowAntagonists
Cat.No. Product Name
0173 (RS)-CPP  
Price and Availability

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(RS)-CPP
Chemical Name: (RS)-3-(2-Carboxypiperazin-4-yl)-propyl-1-phosphonic acid

Biological Activity:

Potent NMDA antagonist. See separate isomer (Cat. No. 0247).

Technical Data:

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M.Wt: 252.21
Formula: C8H17N2O5P
Storage: Desiccate at RT
Solubility: Soluble to 100 mM in Water
CAS No: [100828-16-8]

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    References:

    Davies et al (1986) CPP, a new potent and selective NMDA antagonist. Depression of central neuron responses, affinity for [3H]-D-AP5 binding sites on brain membranes and anti-convulsant activity. Brain Res. 382 169.

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    Keywords: (RS)-CPP, Ligand-gated Ion Channels, Potent NMDA Antagonist, CPP, Tocris Bioscience
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