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Category:
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7TM Receptors Opioid ReceptorsMiscellaneous Opioids
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Cat.No.
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Product Name
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2808 |
Buprenorphine hydrochloride
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Price and Availability
Click here for full price details of
Buprenorphine hydrochloride
Other Information:
This is a controlled substance with associated
conditions of supply; the relevent licence/documentation from the appropriate
governing body will be required.
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Chemical Name:
[5a,7a(S)]-17-(Cyclopropylmethyl)-a-(1,1-dimethylethyl)
-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-a-methyl-6
,14-ethenomorphinan-7-methanol hydrochloride |
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Biological Activity:
ORL1 receptor agonist that also
displays mixed antagonist/partial agonist activity at κ, δ and μ-opioid
receptors.
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Technical Data:
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Resources:
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Certificate of Analysis / MSDS:
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References:
Wnendt et al
(1999) Agonist effect of buprenorphine in a nociceptin/OFQ receptor-triggered
reporter gene assay. Mol.Pharmacol. 56 334. Tzschentke
(2002) Behavioral pharmacology of buprenorphine, with a focus on preclinical
models of reward and addiction. Psychopharmacol. 161 1.
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Keywords: Buprenorphine Hydrochloride, Opioid Receptors, Opioid Receptor Ligand, Tocris Bioscience
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