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Category: 7TM ReceptorsarrowOpioid ReceptorsarrowDelta ReceptorsarrowAntagonists
Cat.No. Product Name
0754 N-Benzylnaltrindole hydrochloride  
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N-Benzylnaltrindole hydrochloride
Chemical Name: 1'-Benzyl-17-(cyclopropylmethyl)-6,7-didehydro-4,5a-epo xy-3,14-dihydroxyindolo[2',3':6,7]morphinan hydrochloride

Biological Activity:

Potent δ2-selective opioid receptor antagonist with a long duration of action in vivo.

Technical Data:

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M.Wt: 541.09
Formula: C33H32N2O3.HCl
Storage: Store at RT
Solubility: Soluble in DMSO

Resources:

  • Certificate of Analysis / MSDS:

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    Product/Material Safety Data Sheet: View current batch
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    References:

    Korlipara et al (1994) N-Benzylnaltrindoles as long acting δ-opioid receptor antagonists. J.Med.Chem. 37 1882.
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    Keywords: N-Benzylnaltrindole Hydrochloride, Opioid Receptors, D2 Selective Non-peptide Antagonist, NBenzylnaltrindole Hydrochloride, Tocris Bioscience

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