BTCP Maleate | Neurotransmitter Transporters | Potent Dopamine Uptake Inhibitor

Category:

Cat.No.	Product Name
0702	BTCP maleate

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BTCP maleate

Chemical Name: 1-[1-(2-Benzo[b]thienyl)cyclohexyl)]piperidine maleate

Biological Activity:

A potent dopamine re-uptake inhibitor with a behavioural profile different from that of PCP and similar to that of cocaine.

Technical Data:

M.Wt:	415.55
Formula:	C₁₉H₂₅NS.C₄H₄O₄
Storage:	Desiccate at +4°C
Solubility:	Soluble to 100 mM in DMSO
Purity:	>98%
CAS No:	[112726-66-6]

Resources:

Certificate of Analysis / MSDS:

Certificate of Analysis: View current batch

Product/Material Safety Data Sheet: View current batch

References:

Vignon et al.(1988) [³H]N-[1-(2-benzo[b]thiophenyl)cyclohexyl]piperidine ([³H]BTCP): a new phencyclidine analogue selective for the dopamine uptake complex. Eur.J.Pharmacol. 148 427. Koek et al (1989) The phencyclidine (PCP) analogue N-[1-(2-benzo(b)thiophenyl)cyclohexyl]piperidine shares cocaine-like but not other characteristic behavioural effects with PCP, ketamine and MK-801. J.Pharmacol.Exp.Ther. 250 1019. Chergui et al (1992) Inhibition of the locus coeruleus neurons by the phenylcyclidine analog, N-[1-(2-benzo(b)thiophenyl)cyclohexyl]-piperidine: evidence for potent indirect adrenoceptor agonist properties. Eur.J.Pharmacol. 219 169.

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Keywords: BTCP Maleate, Neurotransmitter Transporters, Potent Dopamine Uptake Inhibitor, Tocris Bioscience

Literature in this Area

Scientific Reviews

Dopamine Receptors
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Product Feature

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