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Category:
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7TM Receptors Opioid ReceptorsKappa ReceptorsAgonists
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Cat.No.
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Product Name
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0699 |
BRL 52537 hydrochloride
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Price and Availability
Click here for full price details of
BRL 52537 hydrochloride
Other Information:
Sold with the permission of GlaxoSmithKline
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Chemical Name:
(±)-1-(3,4-Dichlorophenyl)acetyl-2-(1-pyrrolidinyl)meth
ylpiperidine hydrochloride |
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Biological Activity:
The most κ/μ-selective and among the most potent κ ligands known (25 times more potent than morphine in vivo).
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Technical Data:
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Resources:
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Certificate of Analysis / MSDS:
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For specific/earlier batch please select:
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References:
Vecchietti et al (1991) (2S)-1-(Arylacetyl)-2-(aminomethyl)piperidine
derivatives: novel, highly selective κ opioid analgesics.
J.Med.Chem. 34 397.
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or by Research Area
Keywords: BRL 52537 Hydrochloride, Opioid Receptors, Potent & Selective K Agonist, BRL52537 Hydrochloride, Tocris Bioscience
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