BIM 23052 | Peptides (Hypothalamic / Pituitary Hormones) | Sst5 Agonist | BIM23052

Category:

Peptides (Hypothalamic/Pituitary Hormones)

Cat.No.	Product Name
2842	BIM 23052

Price and Availability

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BIM 23052

Biological Activity:

Somatostatin sst₅ receptor agonist (K_i values are 7.3, 13.5, 31.3 and 141 nM for sst₅, sst₂, sst₁ and sst₄ receptors respectively). Stimulates gastric emptying following i.c. administration.

Technical Data:

M.Wt:	1122.3
Formula:	C₆₁H₇₅N₁₁O₁₀
Storage:	Store at -20°C
CAS No:	[133073-82-2]

Resources:

Certificate of Analysis / MSDS:

Certificate of Analysis: View current batch

Product/Material Safety Data Sheet: View current batch

References:

Patel and Srikant (1994) Subtype selectivity of peptide analogs for all five cloned human somatostatin receptors (hsstr 1-5). Endocrinol. 135 2814. Martinez et al (2000) Intracisternal injection of somatostatin receptor 5-preferring agonists induces a vagal cholinergic stimulation of gastric emptying in rats. J.Pharmacol.Exp.Ther. 293 1099. Nunn et al (2002) Pharmacological characterisation of the goldfish somatostatin sst₅ receptor. Eur.J.Pharmacol. 436 173.

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Keywords: BIM 23052, Peptides (Hypothalamic / Pituitary Hormones), Sst5 Agonist, BIM23052, Tocris Bioscience

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Product Feature

Somatostatin Receptors

Key somatostatin receptor compounds available from Tocris include:

1980 L-817,818

Potent and selective sst5 agonist

2440 NNC 26-9100

Selective sst4 agonist

1979 L-803,087

Potent and selective sst4 agonist

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