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Category: Ion ChannelsarrowLigand-gated Ion ChannelsarrowGlutamate (Ionotropic) ReceptorsarrowAMPA / Kainate SelectivearrowMiscellaneous
Cat.No. Product Name
0253 (R)-AMPA  
Price and Availability

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(R)-AMPA
Chemical Name: (R)-a-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid

Biological Activity:

Inactive enantiomer of AMPA.

Technical Data:

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M.Wt: 186.17
Formula: C7H10N2O4
Storage: Store at RT
Solubility: Soluble to 10 mM in Water
CAS No: [83654-13 -1]

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    • Certificate of Analysis / MSDS:

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    References:

    Hansen et al (1983) Enzymic resolution and binding to rat brain membranes of the glutamic acid agonist α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid. J.Med.Chem. 26 901. Lauridsen et al (1985) Ibotenic acid analogues. Synthesis, molecular flexibility, and in vitro activity of agonists and antagonists at central glutamic acid receptors. J.Med.Chem. 28 668.
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    Keywords: (R)-AMPA, Ligand-gated Ion Channels, Inactive Isomer Of (RS)-AMPA (0169), AMPA, Tocris Bioscience
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