Home » Pharmacology » Transporters » Neurotransmitter Transporters » Cannabinoid Transporters » OMDM-2

OMDM-2

Cat. No. 1797

Price and Availability

For OMDM-2 pricing & availability please select your country from the drop down menu:
Submit

By clicking submit you agree to accept a cookie from Tocris Bioscience. For details, please read our privacy and cookie policy.

Chemical Name: (9Z)-N-[1-((R)-4-Hydroxbenzyl)-2-hydroxyethyl]-9-octadecenamide

Biological Activity

Metabolically stable inhibitor of anandamide cellular uptake (K_i = 3 μM). Displays relatively low affinity for CB₁ and CB₂ receptors (K_i values are 5.1 and > 10 μM) and for vanilloid VR1 receptors (EC₅₀ = 10 μM). Has minimal activity against FAAH (K_i > 50 μM). Active in vivo.

Technical Data

M.Wt:

431.66

Formula:

C₂₇H₄₅NO₃

Solubility:

Soluble to 10 mM in ethanol and to 10 mM in DMSO

Purity:

>99 %

Storage:

Store at +4°C

CAS No:

616884-63-0

The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.

Resources

Certificate of Analysis / Safety Data Sheet

Certificate of Analysis: View current batch

Safety Data Sheet: View Safety Data Sheet

References

Ortar et al (2003) Novel selective and metabolically stable inhibitors of anandamide cellular uptake. Biochem.Pharmacol. 35 1473. PMID: 12732359.

de Lago et al (2004) In vivo pharmacological actions of two novel inhibitors of anandamide cellular uptake. Eur.J.Pharmacol. 484 249. PMID: 14744610.

If you know of a relevant citation for this product please let us know.