CGS 15943Cat No. 1699 |
Price and Availability |
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Chemical Name: 9-Chloro-2-(2-furanyl)-[1,2,4]triazolo[1,5-c]quinazolin -5-amine |
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Biological Activity
Potent adenosine receptor antagonist (Ki values are 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively). Orally active in vivo.Technical Data
M.Wt:The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis and MSDS.
Resources
Certificate of Analysis / MSDS
References
Williams et al (1987) Biochemical characterization of the triazoloquinazoline CGS 15943, a novel, non-xanthine adenosine antagonist. J.Pharmacol.Exp.Ther. 241 415. Ghai et al (1987) Pharmacological characterization of CGS 15943A: a novel nonxanthine adenosine antagonist. J.Pharmacol.Exp.Ther. 242 784. Klotz (2000) Adenosine receptors and their ligands. Naunyn-Schmied.Arch.Pharmacol. 362 382.If you know of a useful citation for this product please let us know.
Keywords: CGS 15943, Potent, adenosines, receptor, antagonists, Non-Selective, Receptors, CGS15943
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