Cat. No. 1034
Alternative Name: AH 024
Chemical Name: cis-4-Phenyl-2-propionamidotetralin
Biological ActivityMelatonin receptor antagonist, >300-fold selective for the MT2 (vs MT1) subtype.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Dubocovich et al (1995) Melatonin receptors: are there multiple subtypes? TiPS 16 50. PMID: 7762083.
Dubocovich et al (1997) Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroceptor. Naunyn Schmiedebergs Arch.Pharmacol. 355 365. PMID: 9089668.
If you know of a relevant citation for this product please let us know.
View Related Products by Target
View Related Products by Product Action
Keywords: 4-P-PDOT, supplier, MT2, antagonists, Receptors, Melatonin, AH024, Tocris Bioscience, Melatonin Receptor Antagonists
Find multiple products by catalog number
New Products in this Area
Selective S1P2 allosteric agonistMRS 2905
Potent and selective P2Y14 receptor agonistTreprostinil
Potent prostacyclin (PGI2) analogS 18886
Potent thromboxane A2 (TP) antagonist
Follow @Tocris on Twitter
Tocris is now actively tweeting. For regular updates on news, events and special offers, follow @Tocris on Twitter.