R&D Systems Inc. Tocris Bioscience Boston Biochem

4-P-PDOT

Cat. No. 1034

4-P-PDOT C19H21NO [134865-74-0]

Price and Availability

For 4-P-PDOT pricing & availability please select your country from the drop down menu:
Submit
By clicking submit you agree to accept a cookie from Tocris Bioscience. For details, please read our privacy and cookie policy.

Alternative Name: AH 024

Chemical Name: cis-4-Phenyl-2-propionamidotetralin

Biological Activity

Melatonin receptor antagonist, >300-fold selective for the MT2 (vs MT1) subtype.

Technical Data

M.Wt:
279.38
Formula:
C19H21NO
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in ethanol
Purity:
>99 %
Storage:
Store at RT
CAS No:
134865-74-0

The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.

Certificate of Analysis / Safety Data Sheet

Certificate of Analysis: View current batch
Select another batch:
Safety Data Sheet: View Safety Data Sheet

References

Dubocovich et al (1995) Melatonin receptors: are there multiple subtypes? TiPS 16 50. PMID: 7762083.

Dubocovich et al (1997) Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroceptor. Naunyn Schmiedebergs Arch.Pharmacol. 355 365. PMID: 9089668.

If you know of a relevant citation for this product please let us know.

View Related Products by Target

Keywords: 4-P-PDOT, supplier, MT2, antagonists, Receptors, Melatonin, AH024

Quick Order

Find multiple products by catalog number

divider line

New Product E-alerts

Sign up for email updates from Tocris

e-alerts

Enter your email address below to sign up to receive our email updates:

divider line

New Products in this Area

DC 260126

FFA1 (GPR40) antagonist

AR-C 118925XX

Selective, competitive P2Y2 receptor antagonist

NIBR 189

Potent and selective EBI2 (GPR183) receptor antagonist

ONO AE3 208

High affinity and selective EP4 antagonist

TCS 3035

GPR35 agonist

PF 5274857 hydrochloride

Potent and selective Smoothened (Smo) receptor antagonist

GSK 137647

Potent and selective FFA4 (GPR120) agonist

AH 7614

Selective FFA4 (GPR120) antagonist

Sign-up for new product e-alerts
divider line

Bio-Techne Events

Pharmacology 2014

Pharmacology 2014

December 16 - 18, 2014

London, UK

Booth Number: 12