Cat. No. 1034
Alternative Name: AH 024
Chemical Name: cis-4-Phenyl-2-propionamidotetralin
Biological ActivityMelatonin receptor antagonist, >300-fold selective for the MT2 (vs MT1) subtype.
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Certificate of Analysis / Safety Data Sheet
Dubocovich et al (1995) Melatonin receptors: are there multiple subtypes? TiPS 16 50. PMID: 7762083.
Dubocovich et al (1997) Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroceptor. Naunyn Schmiedebergs Arch.Pharmacol. 355 365. PMID: 9089668.
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Keywords: 4-P-PDOT, supplier, MT2, antagonists, Receptors, Melatonin, AH024
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