Cat. No. 3500
Chemical Name: rel-5-(1,1-Dimethylheptyl)-2-[(1R,3
Biological ActivityPotent CB1 receptor agonist (Ki = 2.2 nM). Display 3 - 28-fold > potency than Δ9-THC (Cat. No. 2741). Exhibits analgesic, motor depressant, anticonvulsant and hypothermic effects in vivo.
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Certificate of Analysis / Safety Data Sheet
Weissman et al (1982) Cannabimimetic activity from CP-47,497, a derivative of 3-phenylcyclohexanol. J.Pharmacol.Exp.Ther. 223 516. PMID: 6290642.
Melvin et al (1993) Structure-activity relationships for cannabinoid receptor-binding and analgesic activity: studies of bicyclic cannabinoid analogs. Mol.Pharmacol. 44 1008. PMID: 8246904.
Huffman et al (2008) Synthesis and pharmacology of 1-deoxy analogs of CP-47,497 and CP-55,940. Bioorg.Med.Chem. 16 322. PMID: 17919913.
If you know of a relevant citation for this product please let us know.
Keywords: (±)-CP 47497, supplier, Potent, CB1, agonists, cannabinoids, Receptors, (±)-CP47497, cb1r
Find multiple products by catalog number
New Products in this Area
CB1 receptor negative allosteric modulatorVirodhamine trifluoroacetate
TFA salt of virodhamine, an endogenous cannabinoid receptor mixed agonist/antagonist
March 28 - April 1, 2015