(±)-CP 47497

Cat. No. 3500

()-CP 47497 C21H34O2 [70434-82-1]

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Chemical Name: rel-5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3-hydroxycyclohexyl]phenol

Biological Activity

Potent CB1 receptor agonist (Ki = 2.2 nM). Display 3 - 28-fold > potency than Δ9-THC (Cat. No. 2741). Exhibits analgesic, motor depressant, anticonvulsant and hypothermic effects in vivo.

Technical Data

Soluble to 100 mM in DMSO and to 100 mM in ethanol
>98 %
Store at -20°C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Safety Data Sheet

Certificate of Analysis: View current batch
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Safety Data Sheet: View Safety Data Sheet


Weissman et al (1982) Cannabimimetic activity from CP-47,497, a derivative of 3-phenylcyclohexanol. J.Pharmacol.Exp.Ther. 223 516. PMID: 6290642.

Melvin et al (1993) Structure-activity relationships for cannabinoid receptor-binding and analgesic activity: studies of bicyclic cannabinoid analogs. Mol.Pharmacol. 44 1008. PMID: 8246904.

Huffman et al (2008) Synthesis and pharmacology of 1-deoxy analogs of CP-47,497 and CP-55,940. Bioorg.Med.Chem. 16 322. PMID: 17919913.

If you know of a relevant citation for this product please let us know.

View Related Products by Target

Keywords: ()-CP 47497, supplier, Potent, CB1, agonists, cannabinoids, Receptors, ()-CP47497, cb1r

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