Cat. No. 3500
Chemical Name: rel-5-(1,1-Dimethylheptyl)-2-[(1R,3
Biological ActivityPotent CB1 receptor agonist (Ki = 2.2 nM). Display 3 - 28-fold > potency than Δ9-THC (Cat. No. 2741). Exhibits analgesic, motor depressant, anticonvulsant and hypothermic effects in vivo.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Weissman et al (1982) Cannabimimetic activity from CP-47,497, a derivative of 3-phenylcyclohexanol. J.Pharmacol.Exp.Ther. 223 516. PMID: 6290642.
Melvin et al (1993) Structure-activity relationships for cannabinoid receptor-binding and analgesic activity: studies of bicyclic cannabinoid analogs. Mol.Pharmacol. 44 1008. PMID: 8246904.
Huffman et al (2008) Synthesis and pharmacology of 1-deoxy analogs of CP-47,497 and CP-55,940. Bioorg.Med.Chem. 16 322. PMID: 17919913.
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Keywords: (±)-CP 47497, supplier, Potent, CB1, agonists, cannabinoids, Receptors, (±)-CP47497, cb1r
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