UCPH 101Cat No. 3490 |
Price and Availability |
|
Chemical Name: 2-Amino-5,6,7,8-tetrahydro-4-(4-methoxyphenyl)-7-(napht halen-1-yl)-5-oxo-4H-chromene-3-carbonitrile |
|
Biological Activity
Selective non-substrate inhibitor of EAAT1 (IC50 values are 660, >300000 and >300000 nM for EAAT1, EAAT2 and EAAT3 respectively).Licensing Information
Sold under license from Hugin Neurochemicals.Technical Data
M.Wt:The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis and MSDS.
Resources
Certificate of Analysis / MSDS
References
Jensen et al (2009) Discovery of the first selective inhibitor of excitatory amino acid transporter subtype 1. J.Med.Chem. 52 912. Bunch et al (2009) Excitatory amino acid transporters as potential drug targets. Exp.Opin.Ther.Targets 13 719.If you know of a useful citation for this product please let us know.
Keywords: UCPH 101, Selective, non-substrate, EAAT1, inhibitors, excitatory, amino, acid, transporters, glutamate, monoamine, neurotransmitter, GLAST
Buy Now / Print Quote
Find multiple products by catalog number
Print Quote Facility
Order via your purchasing department
It's now even easier to place orders via your purchasing department.
Simply add a product to your cart & click on the "Print Quote" button.
Calcium Imbalance and Neuroprotective Targets
Written by E. Besancon et al
'Calcium Imbalance and Neuro-protective Targets in Cerebral Ischemia & Brain Injury' highlights the key targets involved in stroke, trauma and neurodegeneration.
RSS News Feed
Find out about new products as soon as they go live!
Click on the orange RSS button to read more about our RSS feed and actively opt in.