Fentanyl citrateCat No. 3247 |
Price and Availability |
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Alternative Name: Phentanylcitrate Chemical Name: N-Phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]propanamide citrate |
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Biological Activity
Potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively). Displays antinociceptive activity in vivo.Technical Data
M.Wt:The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis and MSDS.
Resources
Certificate of Analysis / MSDS
References
Zernig et al (1995) Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding. Life Sci. 57 2113. Liu et al (2003) Opioid activity of C8813, a novel and potent opioid analgesic. Life Sci. 73 233. Stevenson et al (2003) Opioid interactions in rhesus monkeys: effects of d + m and d + k agonists on schedule-controlled responding and thermal nociception. J.Pharmacol.Exp.Ther. 307 1054.If you know of a useful citation for this product please let us know.
Keywords: Fentanyl citrate, Potent, selective, μ-opioid, mu-opioid, agonists, MOP, Receptors, OP3
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