R&D Systems Inc. Tocris Bioscience Boston Biochem

Sulprostone

Cat. No. 3049

Sulprostone C23H31NO7S [60325-46-4]

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Chemical Name: (5Z)-7-[(1R,2R,3R)-3-Hydroxy-2-[(1E,3R)-3-hydroxy-4-buten-1-yl]-5-oxocyclopentyl]-N-(methylsulfonyl)-5-heptenamide

Biological Activity

Selective EP3 and EP1 receptor agonist (Ki values are 0.6 and 21 nM respectively). Synthetic PGE2 analog and allodynic agent.

Technical Data

M.Wt:
465.56
Formula:
C23H31NO7S
Solubility:
Soluble in methyl acetate (supplied pre-dissolved -10mg/ml)
Storage:
Store at -20°C
CAS No:
60325-46-4

The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.

Certificate of Analysis / Safety Data Sheet

Certificate of Analysis: View current batch
Safety Data Sheet: View Safety Data Sheet

References

Narumiya et al (1999) Prostanoid receptors: Structures, properties, and functions. Phys.Rev. 79 1193.

Gil et al (2008) Transient allodynia pain models in mice for assessment of analgesic activity. Br.J.Pharmacol. 153 769. PMID: 17700719.

If you know of a relevant citation for this product please let us know.

View Related Products by Target

Keywords: Sulprostone, supplier, Sulprostone, prostaglandin, prostanoid, EP1, EP3, receptor, agonist

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