Cat. No. 3049
Chemical Name: (5Z)-7-[(1R,2R,3R)-3-Hydroxy-2-[(1E
Biological ActivitySelective EP3 and EP1 receptor agonist (Ki values are 0.6 and 21 nM respectively). Synthetic PGE2 analog and allodynic agent.
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Certificate of Analysis / Safety Data Sheet
Narumiya et al (1999) Prostanoid receptors: Structures, properties, and functions. Phys.Rev. 79 1193.
Gil et al (2008) Transient allodynia pain models in mice for assessment of analgesic activity. Br.J.Pharmacol. 153 769. PMID: 17700719.
If you know of a relevant citation for this product please let us know.
View Related Products by Target
Keywords: Sulprostone, supplier, Sulprostone, prostaglandin, prostanoid, EP1, EP3, receptor, agonist
Find multiple products by catalog number
New Products in this Area
High affinity and selective EP4 antagonistTCS 3035
GPR35 agonistPF 5274857 hydrochloride
Potent and selective smoothened (Smo) receptor antagonistGSK 137647
Potent and selective FFA4 (GPR120) agonistAH 7614
Selective FFA4 (GPR120) antagonistProsaptide TX14(A)
Potent GPR37 and GPR37L1 agonist
Follow @Tocris on Twitter
Tocris is now actively tweeting. For regular updates on news, events and special offers, follow @Tocris on Twitter.