Cat. No. 3049
Chemical Name: (5Z)-7-[(1R,2R,3R)-3-Hydroxy-2-[(1E
Biological ActivitySelective EP3 and EP1 receptor agonist (Ki values are 0.6 and 21 nM respectively). Synthetic PGE2 analog and allodynic agent.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Narumiya et al (1999) Prostanoid receptors: Structures, properties, and functions. Phys.Rev. 79 1193.
Gil et al (2008) Transient allodynia pain models in mice for assessment of analgesic activity. Br.J.Pharmacol. 153 769. PMID: 17700719.
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Keywords: Sulprostone, supplier, Sulprostone, prostaglandin, prostanoid, EP1, EP3, receptor, agonist
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March 14 - 18, 2015