Cat. No. 3049
Chemical Name: (5Z)-7-[(1R,2R,3R)-3-Hydroxy-2-[(1E
Biological ActivitySelective EP3 and EP1 receptor agonist (Ki values are 0.6 and 21 nM respectively). Synthetic PGE2 analog and allodynic agent.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Narumiya et al (1999) Prostanoid receptors: Structures, properties, and functions. Phys.Rev. 79 1193.
Gil et al (2008) Transient allodynia pain models in mice for assessment of analgesic activity. Br.J.Pharmacol. 153 769. PMID: 17700719.
If you know of a relevant citation for this product please let us know.
View Related Products by Target
Keywords: Sulprostone, supplier, Sulprostone, prostaglandin, prostanoid, EP1, EP3, receptor, agonist
Find multiple products by catalog number
New Products in this Area
P2Y12 inhibitorRactopamine hydrochloride
Trace amine 1 (TA1) receptor agonistTG 4-155
High affinity and selective EP2 receptor antagonistSAG
Potent Smoothened receptor agonist; activates the Hedgehog signaling pathwayDC 260126
FFA1 (GPR40) antagonistAR-C 118925XX
Selective, competitive P2Y2 receptor antagonistEPPTB
Trace amine 1 (TA1) receptor antagonist/inverse agonistNIBR 189
Potent and selective EBI2 (GPR183) receptor antagonistONO AE3 208
High affinity and selective EP4 antagonist
April 12 - 15, 2015