DiprenorphineCat No. 2965 |
Price and Availability |
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Chemical Name: 17-(Cyclopropylmethyl)-4,5-epoxy-18,19-dihydro-3-hydrox y-6-methoxy-a,a-dimethyl-6,14-ethenomorphinan-7-methano l |
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Biological Activity
Non-selective opioid receptor antagonist (Ki values are 0.017, 0.072 and 0.23 nM for κ-, μ- and δ-opioid receptors).Technical Data
M.Wt:The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis and MSDS.
Resources
Certificate of Analysis / MSDS
References
Paterson et al (1983) Classification of opioid receptors. Br.Med.Bull. 39 31. Raynor et al (1994) Pharmacological characterization of the cloned k-, d-, and m-opioid receptors. Mol.Pharmacol. 45 330. Iwasaki et al (1994) The effect of the nonselective opioid antagonist diprenorphine vasopressin secretion in the rat. Endocrinology 134 48.If you know of a useful citation for this product please let us know.
Keywords: Diprenorphine, Non-Selective, opioids, antagonists, Receptors
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