Naloxonazine dihydrochloride

Cat. No. 0591

Naloxonazine dihydrochloride C38H42N4O6.2HCl [880759-65-9]

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Chemical Name: Bis-[5-α-4,5-Epoxy-3,14-dihydroxy-17-(2-propenyl)-morphinan-6-ylidene] hydrazine dihydrochloride

Biological Activity

Potent opioid antagonist, selective for μ1 receptors.

Technical Data

Soluble to 25 mM in water
>98 %
Store at RT

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Safety Data Sheet

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Paul et al (1988) Differential blockade by naloxonazine of two μ opiate actions: analgesic and inhibition of gastrointestinal transit. Eur.J.Pharmacol. 149 403. PMID: 2842168.

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Keywords: Naloxonazine dihydrochloride, supplier, Selective, antagonists, μ-opioid, mu-opioid, μ1-opioid, mu1-opioid, MOP, Receptors, OP3, μ Opioid Receptor Antagonists

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