Zinterol hydrochlorideCat No. 1051 |
Price and Availability |
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Alternative Name: MJ 9184 Chemical Name: N-[5-[2-[(1,1-Dimethyl-2-phenylethyl)amino]-1-hydroxyet hyl]-2-hydroxyphenyl]methanesulphonamide hydrochloride |
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Biological Activity
Potent and selective β2-adrenoceptor agonist (pKB values are 8.3 and < 5.7 for β 2 and β1 receptors respectively, as measured in human artery).Technical Data
M.Wt:The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis and MSDS.
Resources
Certificate of Analysis / MSDS
References
Kaumann (1997) Four b-adrenoceptor subtypes in the mammalian heart. TiPS 18 70. Arvydas Skeberdis et al (1997) Beta-2 adrenergic activation of L-type Ca2+ current in cardiac myocytes. J.Pharmacol.Exp.Ther. 283 452. Hutchinson et al (2006) Agonist effects of zinterol at the mouse and human b3-adrenoceptor. Naunyn-Schmied.Arch.Pharmacol. 373 158.If you know of a useful citation for this product please let us know.
Keywords: Zinterol hydrochloride, Selective, α2-adrenoceptor, beta2-adrenoceptor, b2-adrenoceptor, β2-adrenergic, α2-adrenergic, beta2-adrenergic, b2-adrenergic, agonists, Receptors, MJ9184
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