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IPAGCat. No. 0544 |
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Chemical Name: 1-(4-Iodophenyl)-3-(2-adamantyl)guanidine |
Biological Activity
Potent σ-receptor antagonist.Certificate of Analysis / Safety Data Sheet
Certificate of Analysis: View current batch
Safety Data Sheet: View Safety Data Sheet
References
Wilson et al (1991) Radiosynthesis of σ receptor ligands for positron emission tomography: 11C- and 18F-labelled guanidines. J.Med.Chem. 34 1867. PMID: 1648140.
Whittemore et al (1997) Antagonism of N-methyl-D-aspartate receptors by σ site ligands: potency, subtype-selectivity and mechanisms of inhibition. J.Pharmacol.Exp.Ther. 282 326. PMID: 9223571.
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Keywords: IPAG, supplier, Potent, σ, sigma, antagonists, General, Receptors
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