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L-759,656Cat. No. 2434 |
Price and Availability |
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Chemical Name: (6aR,10aR)-3-(1,1-Dimethylheptyl)-6 |
Biological Activity
Highly selective CB2 receptor agonist (Ki values are 11.8 and 4888 nM for CB2 and CB1 receptors respectively). Potently inhibits forskolin-stimulated cAMP production via CB2 receptors expressed in CHO cells (EC50 = 3.1 nM).Certificate of Analysis / Safety Data Sheet
References
Ross et al (1999) Agonist-inverse agonist characterization at CB1 and CB2 cannabinoid receptors of L759633, L759656 and AM630. Br.J.Pharmacol. 126 665. PMID: 10188977.
Huffman (2000) The search for selective ligands for the CB2 receptor. Curr.Pharmaceut.Des. 6 1323.
Huffman (2005) CB2 receptor ligands. Mini Rev.Med.Chem. 5 641. PMID: 16026310.
If you know of a relevant citation for this product please let us know.
Keywords: L-759,656, Supplier, selective, CB2, agonists, cannabinoids, Receptors, cb2r, L759656
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