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DPPE fumarateCat. No. 0743 |
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Chemical Name: N,N-Diethyl-2-[4-(phenylmethyl)phenoxy]ethanamine fumarate |
Biological Activity
Binds with high affinity to the antiestrogen binding site but not to the estrogen receptor. An inhibitor of histamine binding at the intracellular histamine (Hlc) site.Technical Data
M.Wt:The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Certificate of Analysis / Safety Data Sheet
References
Brandes and Hermonat (1984) A diphenylmethane derivative specific for the antiestrogen binding site found in rat liver microsomes. Biochem.Biophys.Res.Commun. 123 724. PMID: 6548377.
Brandes et al (1990) Histamine as an intracellular messenger. Biochem.Pharmacol. 40 1677. PMID: 2242003.
Sturman et al (1994) Modulation of the intracellular and H3-histamine receptors and chemically-induced seizures in mice. Agents Actions 41 C68. PMID: 7976808.
If you know of a relevant citation for this product please let us know.
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Keywords: DPPE fumarate, supplier, Ligand, antiestrogen, binding, site, inhibitors, histamine, intracellular, ER, ERR, Estrogen, Receptors, Histaminergic-, Compounds
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