Carcinine ditrifluoroacetateCat No. 2211 |
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Chemical Name: 3-Amino-N-[2-(1H-imidazol-4-yl)ethyl]propanamide ditrifluoroacetate |
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Biological Activity
Highly selective H3 receptor antagonist (Ki values are 0.30, 365 and 3621 μM for H3, H2 and H1 receptors respectively). Acts as a natural antioxidant with hydroxyl radical scavenging and lipid peroxidase activities.Technical Data
M.Wt:The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis and MSDS.
Resources
Certificate of Analysis / MSDS
References
Babizhayev et al (1994) L-Carnosine (b-alanyl-L-histidine) and carcinine (b-alanylhistamine) act as natural antioxidants with hydroxyl-radical-scavenging and lipid-peroxidase activities. Biochem.J. 304 509. Chen et al (2004) Pharmacological effects of carcinine on histaminergic neurons in the brain. Br.J.Pharmacol. 143 573.If you know of a useful citation for this product please let us know.
Keywords: Carcinine ditrifluoroacetate, Highly, selective, H3, antagonists, Histamine, H3, Receptors, histaminergic
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