More Information »Vanilloids are a group of compounds, structurally related to capsaicin, thought to exert their actions via vanilloid receptors. The vanilloid receptor family (TRPV) is a member of the transient receptor potential (TRP) superfamily of ion channels, and have six members (TRPV1-6).

TRPV Products

Product Name / Activity
1116 AM 404
Vanilloid receptor agonist. Also anandamide transport inhibitor
1339 Anandamide
Endogenous CB and TRPV1 receptor agonist
1017 Anandamide (in Tocrisolve™ 100)
Endogenous CB and TRPV1 receptor agonist (in water-soluble emulsion)
1354 Arvanil
Potent TRPV1 (VR1) and CB1 agonist/anandamide transport inhibitor
0462 (E)-Capsaicin
Prototypic vanilloid receptor agonist
1556 6'-Iodoresiniferatoxin
High affinity TRPV1 agonist/partial agonist
1568 NADA
Endogenous TRPV1 agonist. Also CB1 agonist
1641 OLDA
Potent, selective endogenous TRPV1 agonist
0934 Olvanil
Potent vanilloid receptor agonist
1466 PPAHV
Non-pungent vanilloid receptor agonist
1137 Resiniferatoxin
Potent vanilloid receptor agonist
3745 RN 1747
Selective TRPV4 agonist
Product Name / Activity
5781 A 425619
Potent TRPV1 antagonist
4319 A 784168
Potent and selective TRPV1 antagonist
4330 AMG 21629
Potent and selective TRPV1 antagonist
5995 AMG 517
Potent TRPV1 antagonist
2316 AMG 9810
Potent and selective, competitive antagonist of TRPV1
2836 Arachidonyl serotonin
Dual FAAH inhibitor/TRPV1 antagonist
3875 BCTC
TRPV1 antagonist
0464 Capsazepine
Vanilloid receptor antagonist; also activator of ENaCδ
5106 GSK 2193874
Potent and selective TRPV4 antagonist; orally active
4100 HC 067047
Potent and selective TRPV4 antagonist
1975 6-Iodonordihydrocapsaicin
Potent, competitive vanilloid receptor antagonist
1362 5'-Iodoresiniferatoxin
Potent, silent TRPV1 antagonist
3361 JNJ 17203212
Reversible, competitive and potent TRPV1 antagonist
1577 L-R4W2
TRPV1 antagonist peptide
3746 RN 1734
Selective TRPV4 antagonist
5678 RN 9893 hydrochloride
Potent and selective TRPV4 antagonist
1439 Ruthenium Red
Blocks capsaicin-activated cation channels
1615 SB 366791
Potent, selective, competitive TRPV1 antagonist
3265 SB 452533
Potent TRPV1 receptor antagonist
4729 α-Spinasterol
TRPV1 antagonist; active in vivo
1098 Tranilast
Antiallergic; inhibits TRPV2-mediated responses
Product Name / Activity
5246 MRS 1477
TRPV1 positive allosteric modulator
Ligand Sets
Product Name / Activity
2181 Vanilloid TRPV1 Receptor Tocriset™
Selection of 5 vanilloid TRPV1 receptor ligands (Cat. Nos. 0462, 0934, 1137, 0464 and 1615)
Product Name / Activity
5464 AC 4
Photoswitchable TRPV1 channel blocker
4104 MM-22
Biotinylated anandamide analog; blocks anandamide uptake
2203 PALDA
Endogenous lipid; potentiates effects of endovanilloids at TRPV1 receptors
Endogenous lipid, active in vivo. Enhances effects of endovanilloids at TRPV1 receptors
1684 Tocrisolve™ 100
Water-soluble emulsion; negative control for reagents in TocrisolveTM 100
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