5-HT7 Receptors

More Information »Serotonin 5-HT7 receptors are located primarily in the thalamus, hypothalamus and hippocampus. The function of these receptors includes the regulation of circadian rhythms, thermoregulation, learning and memory and smooth muscle relaxation.

5-HT7 Receptor Products

Agonists
Cat.No.
Product Name / Activity
1968 AS 19
Potent 5-HT7 agonist
2925 LP 12 hydrochloride
5-HT7 agonist
2534 LP 44
High affinity 5-HT7 agonist
Antagonists
Cat.No.
Product Name / Activity
5005 DR 4485 hydrochloride
High affinity and selective 5-HT7 antagonist; orally bioavailable
1523 LY 215840
5-HT2/5-HT7 antagonist
2726 SB 258719 hydrochloride
Selective 5-HT7 antagonist
1612 SB 269970 hydrochloride
Potent and selective 5-HT7 antagonist; brain penetrant
Other
Cat.No.
Product Name / Activity
0458 5-Carboxamidotryptamine maleate
Has high affinity for 5-ht5A and 5-HT7. Also 5-HT1 agonist
0529 8-Hydroxy-DPAT hydrobromide
Has moderate affinity for 5-HT7; also 5-HT1A agonist
4704 LP 20 hydrochloride
Selective 5-HT7 ligand
0590 Metergoline
Has moderate affinity for 5-HT6 and high affinity for 5-HT7. Also 5-HT1/5-HT2 antagonist
0937 Pimozide
High affinity for 5-HT7. Also D2 antagonist
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