Histamine H2 Receptors

More Information »Histamine H2 receptors are Gαs-protein-coupled receptors involved in the suppressive activities of histamine. H2 receptors exhibit a widespread distribution and are found in the gastrointestinal tract, the central nervous system, smooth muscle cells and endothelial cells.

Histamine H2 Receptor Products

Agonists
Cat.No.
Product Name / Activity
0668 Amthamine dihydrobromide
Highly selective standard H2 agonist
0506 Dimaprit dihydrochloride
Standard H2 selective agonist
3545 Histamine dihydrochloride
Endogenous histamine receptor agonist
0646 HTMT dimaleate
H2 / H1 agonist
Antagonists
Cat.No.
Product Name / Activity
0721 Aminopotentidine
H2 antagonist
0902 Cimetidine
H2 antagonist, I1 agonist
0833 ICI 162,846
Potent H2 antagonist, active in vivo
1967 Ranitidine hydrochloride
Selective H2 antagonist
0826 Tiotidine
Potent, selective H2 antagonist
1070 Zolantidine dimaleate
Potent, centrally active H2 antagonist
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