GABAA-ρ Receptors

More Information »GABAA-ρ receptors, previously known as GABAC receptors, are Cys-loop ionotropic ligand-gated ion channels mediating the fast synaptic inhibitory effects of GABA. Despite differing in pharmacology, physiology and biochemistry, they are viewed as a subclass of GABAA receptors.

GABAA-ρ Receptor Products

Agonists
Cat.No.
Product Name / Activity
3618 Acamprosate calcium
GABA agonist and glutamatergic modulator
0344 GABA
Endogenous agonist
0289 Muscimol
Partial GABAA-ρ agonist
4709 RuBi GABA trimethylphosphine
Caged GABA; inhibits neural activity
0181 TACA
GABAA-ρ agonist
Antagonists
Cat.No.
Product Name / Activity
0379 SKF 97541
GABAA-ρ antagonist. Also potent GABAB agonist
0807 THIP hydrochloride
GABAA-ρ antagonist
1040 TPMPA
Selective GABAA-ρ antagonist
0180 ZAPA sulfate
GABAA-ρ antagonist
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