GABAA Receptor Benzodiazepines

Product Name / Activity
5281 AC 5216
Selective TSPO ligand
3568 Bretazenil
Benzodiazepine partial agonist
0405 β-CCB
Benzodiazepine inverse agonist, putative endogenous ligand
2467 CGS 20625
Selective central benzodiazepine receptor partial agonist
0456 Chlormezanone
Skeletal muscle relaxant
1709 CL 218872
Benzodiazepine agonist
2805 Diazepam
Acts at the benzodiazepine modulatory site
0505 Dihydroergotoxine mesylate
Binds to GABAA receptor Cl- channel; allosteric modulator of benzodiazepine site
3083 DMCM hydrochloride
Benzodiazepine inverse agonist
0554 FG 7142
Benzodiazepine inverse agonist
0658 FGIN-1-27
Potent, specific ligand for mitochondrial DBI receptor
0659 FGIN-1-43
Potent, specific ligand for mitochondrial DBI receptor
1328 Flumazenil
Benzodiazepine antagonist
4047 Flunitrazepam
Acts at the benzodiazepene modulatory site
2174 Hispidulin
Partial positive allosteric modulator at the benzodiazepine receptor
1327 L-655,708
Benzodiazepine inverse agonist; selective for α5-containing GABAA receptors
3087 Lorazepam
Acts at the benzodiazepine modulatory site
2832 Midazolam hydrochloride
Benzodiazepine agonist
0670 PK 11195
Antagonist at peripheral benzodiazepine receptors
1997 Ro 15-4513
Benzodiazepine partial inverse agonist
1995 Ro 19-4603
Benzodiazepine inverse agonist
3942 TCS 1105
GABAA α2 benzodiazepine receptor agonist
3655 Zaleplon
Benzodiazepine site agonist
1994 ZK 93423 hydrochloride
Potent benzodiazepine agonist
1996 ZK 93426 hydrochloride
Potent, competitive benzodiazepine antagonist
0655 Zolpidem
Benzodiazepine agonist
1094 Zopiclone
Benzodiazepine agonist

View all GABAA Receptor products

Quick Order

Find multiple products by catalog number

divider line

Pain Research Product Guide

Pain Research Product Guide

Our Pain guide highlights over 280 products for Pain research. Request copy or view PDF today.

divider line

GABA Review

Written by I. Martin et al

GABA Receptors Scientific Review

Our GABA review gives an overview of the structure and function of the GABA receptors, as well as highlighting pharmacological ligands for their study. Request copy or view PDF today.

divider line

Peripheral Sensitization

Written by Grant D. Nicol and Michael R. Vasko

Pain Life Science Poster

Our Peripheral Sensitization poster gives a summary of the excitatory and inhibitory signaling pathways involved in modulation of peripheral sensitization. Request copy or view PDF today.

divider line

Therapeutic Strategies in Schizophrenia

Written by J. Lieberman

Schizophrenia Life Science Poster

Our Schizophrenia poster higlights the targets and pathways representing the most promising strategies to pursue for novel drug development. Request copy today.

divider line

Mechanisms of Addiction

Addiction Life Science Poster

Written by Prof David Nutt, this poster summarizes the brain circuits and neurotransmitter systems that are affected by the main classes of addictive drugs. Request copy or view PDF today.

divider line

Twitter Updates

Follow @Tocris on Twitter

Follow us on Twitter!

Tocris is now actively tweeting. For regular updates on news, events and special offers, follow @Tocris on Twitter.