Adrenergic β3 Receptors

More Information »The adrenergic β3 receptor (β3-adrenoceptor) is a member of the adrenergic receptor group of G-protein-coupled receptors that also includes α1A, α1B, α1D, α2A, α2B, α2C, β1 and β2. They are located primarily in the small intestine, adipose tissue and vascular endothelium.

Adrenergic β3 Receptor Products

Agonists
Cat.No.
Product Name / Activity
0948 BRL 37344, sodium salt
β3 agonist
1134 CGP 12177 hydrochloride
β3 partial agonist. β1/β2 antagonist.
1499 CL 316243 disodium salt
Highly selective β3 agonist
0929 ICI 215,001 hydrochloride
β3 agonist
2197 L-755,507
Very potent and selective β3 partial agonist
2242 Octopamine hydrochloride
Invertebrate biogenic amine: activates β3 adrenoceptors
0994 Pindolol
β3 partial agonist
1060 (S)-(-)-Pindolol
β3 partial agonist. More active enantiomer of pindolol (Cat. No. 0994)
3986 SR 58611A hydrochloride
β3 agonist; displays anxiolytic and antidepressant effects
2154 ZD 2079
β3-adrenoceptor agonist
0930 ZD 7114 hydrochloride
β3 agonist
Antagonists
Cat.No.
Product Name / Activity
2760 L-748,337
Selective β3 antagonist
1511 SR 59230A hydrochloride
Potent and selective β3 antagonist
Ligand Sets
Cat.No.
Product Name / Activity
1873 β-Adrenoceptor Agonist Tocriset™
Selection of 3 β-adrenoceptor agonists (Cat. Nos. 0948, 1747 and 1660)
1874 β-Adrenoceptor Antagonist Tocriset™
Selection of 3 β-adrenoceptor antagonists (Cat. Nos. 1024, 0821 and 1511)
Related Categories

Quick Order

Find multiple products by catalog number

divider line

GPCR Product Listing

GPCR Product Listing

Highlights over 450 products for GPCRs Request copy or view PDF today.

divider line

Cardiovascular Research Product Guide

Cardiovascular Research Product Guide

Our Cardiovascular Guide highlights over 250 products for cardiovascular research. Request copy or view PDF today.

divider line

Regulation of Vascular Reactivity by GPCRs

Written by J.J. Maguire and A.P. Davenport

Cardiovascular Life Science Poster

Our Cardiovascular poster highlights the key G protein-coupled receptors involved in the regulation of vascular reactivity. Request copy today.

divider line

Antidepressants - Current and Future Targets

Written by P. Skolnich et al

Depression Life Science Poster

Our Depression poster highlights presynaptic and postsynaptic targets for the potential treatment of major depressive disorder. Request copy or view PDF today.

divider line

Bio-Techne Events

Neuroscience 2016

Neuroscience 2016

November 12 - 16, 2016

San Diego, CA, USA

Booth: 3217