Adrenergic β1 Receptors

More Information »The adrenergic β1 receptor (β1-adrenoceptor) is a member of the adrenergic receptor group of G-protein-coupled receptors that also includes α1A, α1B, α1D, α2A, α2B, α2C, β2 and β3. They are located primarily in the CNS, heart, coronary artery, kidney and muscle.

Adrenergic β1 Receptors Products

Agonists
Cat.No.
Product Name / Activity
0950 Xamoterol hemifumarate
β1 selective partial agonist
Antagonists
Cat.No.
Product Name / Activity
0387 (RS)-Atenolol
β1 antagonist
0393 (S)-(-)-Atenolol
β1-antagonist. Active isomer of atenolol (Cat. No. 0387)
0906 Betaxolol hydrochloride
Selective β1 antagonist
0914 (±)-Bisoprolol hemifumarate
β1 antagonist
1024 CGP 20712 dihydrochloride
Highly potent and selective β1 antagonist
3256 Metoprolol tartrate
Selective β1 antagonist
3517 Nebivolol hydrochloride
Highly selective β1-adrenoceptor antagonist
0649 (S)-Timolol maleate
β1 antagonist
Ligand Sets
Cat.No.
Product Name / Activity
1874 β-Adrenoceptor Antagonist Tocriset™
Selection of 3 β-adrenoceptor antagonists (Cat. Nos. 1024, 0821 and 1511)
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