Adrenergic β1 Receptors

More Information »The adrenergic β1 receptor (β1-adrenoceptor) is a member of the adrenergic receptor group of G-protein-coupled receptors that also includes α1A, α1B, α1D, α2A, α2B, α2C, β2 and β3. They are located primarily in the CNS, heart, coronary artery, kidney and muscle.

Adrenergic β1 Receptor Products

Agonists
Cat.No.
Product Name / Activity
0950 Xamoterol hemifumarate
β1 selective partial agonist
Antagonists
Cat.No.
Product Name / Activity
0387 (RS)-Atenolol
β1 antagonist
0393 (S)-(-)-Atenolol
β1-antagonist. Active isomer of atenolol (Cat. No. 0387)
0906 Betaxolol hydrochloride
Selective β1 antagonist
0914 (±)-Bisoprolol hemifumarate
β1 antagonist
1024 CGP 20712 dihydrochloride
Highly potent and selective β1 antagonist
3256 Metoprolol tartrate
Selective β1 antagonist
3517 Nebivolol hydrochloride
Highly selective β1-adrenoceptor antagonist
0649 (S)-Timolol maleate
β1 antagonist
Ligand Sets
Cat.No.
Product Name / Activity
1874 β-Adrenoceptor Antagonist Tocriset™
Selection of 3 β-adrenoceptor antagonists (Cat. Nos. 1024, 0821 and 1511)
Related Categories

Quick Order

Find multiple products by catalog number

divider line

Cardiovascular Research Product Guide

Cardiovascular Research Product Guide

Our Cardiovascular Guide highlights over 250 products for cardiovascular research. Request copy or view PDF today.

divider line

GPCR Product Listing

GPCR Product Listing

Highlights over 450 products for GPCRs Request copy or view PDF today.

divider line

Regulation of Vascular Reactivity by GPCRs

Written by J.J. Maguire and A.P. Davenport

Cardiovascular Life Science Poster

Our Cardiovascular poster highlights the key G protein-coupled receptors involved in the regulation of vascular reactivity. Request copy today.

divider line

Antidepressants - Current and Future Targets

Written by P. Skolnich et al

Depression Life Science Poster

Our Depression poster highlights presynaptic and postsynaptic targets for the potential treatment of major depressive disorder. Request copy or view PDF today.

divider line

Bio-Techne Events

Neuroscience 2016

Neuroscience 2016

November 12 - 16, 2016

San Diego, CA, USA

Booth: 3217