5-HT2B Receptors

More Information »Serotonin 5-HT2B receptors, previously known as 5-HT2F receptors, are located primarily in the stomach fundus, uterus, vascular endothelial and vascular and GI smooth muscle, with limited distribution in the brain. 5-HT2B overexpression leads to ventricular hypertrophy.

5-HT2B Receptor Products

Product Name / Activity
1059 BW 723C86 hydrochloride
5-HT2B agonist
0875 m-CPP hydrochloride
5-HT2B/2C receptor agonist
0557 α-Methyl-5-hydroxytryptamine maleate
5-HT2B agonist
Product Name / Activity
3346 ATC 0175 hydrochloride
MCH1 antagonist; also 5-HT2B antagonist and 5-HT1A partial agonist
4081 LY 266097 hydrochloride
Selective 5-HT2B receptor antagonist
3077 LY 272015 hydrochloride
High affinity 5-HT2B antagonist; orally active
2993 RS 127445 hydrochloride
Selective, high affinity 5-HT2B antagonist
1371 SB 200646 hydrochloride
5-HT2C/2B antagonist
1372 SB 204741
Potent, selective 5-HT2B antagonist
1661 SB 206553 hydrochloride
Potent, selective 5-HT2C/5-HT2B antagonist. Orally active
1374 SB 215505
5-HT2B/2C antagonist
1379 SB 221284
Potent, selective 5-HT2C/2B antagonist
1375 SB 228357
5-HT2C/2B antagonist/inverse agonist
1255 SDZ SER 082 fumarate
Selective 5-HT2B/2C antagonist
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