cis MZ 1
Cat. No. 6155
Chemical Name: (2S,4S)-1-((S)-2-(tert-butyl)-17-((
Biological ActivityNegative Control for MZ1 (Cat.No. 6154). Exhibits no significant VHL binding affinity.
Licensing InformationSold under licence from the University of Dundee
External Portal InformationChemicalprobes.org is a portal that offers independent guidance on the selection and/or application of small molecules for research. The use of MZ 1 is reviewed on the chemical probes website.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Zengerle et al (2015) Selective small molecule induced degradation of the BET bromodomain protein BRD4. ACS.Chem.Biol. 10 1770. PMID: 26035625.
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Keywords: cis MZ 1, supplier, cis, MZ1, MZ1, PROTAC, Proteolysis, targeted, chimeras, Bromodomain, BRD2, BRD3, BRD4, BET, proteins, JQ1, VHL, E3, ubiquitin, ligase, HIF-alpha, HIF-a, HIF-α, Tocris Bioscience, Ubiquitin E3 Ligase products
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