Cat. No. 2678
Chemical Name: N-Cyclohexyl-1-(2,4-dichlorophenyl)
Biological ActivitySelective CB2 receptor agonist; Ki values are 7.6 and 900 nM for CB2 and CB1 receptors respectively. Increases P-ERK1/2 expression in HL-60 cells in vitro.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Murineddu et al (2006) Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2',4'-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide. J.Med.Chem. 49 7502. PMID: 17149879.
If you know of a relevant reference for this product please let us know.
Citations are publications that use Tocris products.
Do you know of a great paper that uses GP 2a from Tocris? If so please let us know.
View Related Products by Target
View Related Products by Product Action
Keywords: GP 2a, supplier, Selective, CB2, agonists, cannabinoids, Receptors, GP2a, cb2r, Tocris Bioscience, CB2 Receptor Agonist products