Cat. No. 2678
Chemical Name: N-Cyclohexyl-1-(2,4-dichlorophenyl)
Biological ActivitySelective CB2 receptor agonist; Ki values are 7.6 and 900 nM for CB2 and CB1 receptors respectively. Increases P-ERK1/2 expression in HL-60 cells in vitro.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Murineddu et al (2006) Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2',4'-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide. J.Med.Chem. 49 7502. PMID: 17149879.
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Keywords: GP 2a, supplier, Selective, CB2, agonists, cannabinoids, Receptors, GP2a, cb2r, Tocris Bioscience, CB2 Receptor Agonist products
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Potent and selective CB2 partial agonist; orally biovailable
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