Cat. No. 6033
Chemical Name: N-[(Phenylmethoxy)carbonyl]-L-leucy
Biological ActivityPotent 20S proteasome inhibitor (IC50 = 0.22 nM). Exhibits cytostatic and cytotoxic effects in tumor cells in vitro.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Data Sheet
Mroczkiewicz et al (2010) Studies of the synthesis of all stereoisomers of MG-132 proteasome inhibitors in the tumor targeting approach. J.Med.Chem. 53 1509. PMID: 20112914.
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Keywords: (R)-MG 132, supplier, (R)-MG132, 20S, proteasome, inhibitors, inhibits, potent, Tocris Bioscience, Proteasome Inhibitor products
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