Cat. No. 5965
Chemical Name: 4-(2-Furanyl)-4,10-dihydro-2-methyl
Biological ActivityHigh affinity A2B receptor antagonist (Ki = 3.49 nM). Exhibits >1000-fold selectivity for A2B over A1, A2A and A3 receptors.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Data Sheet
El Maatougui et al (2016) Discovery of potent and highly selective A2B adenosine receptor antagonist chemotypes. J.Med.Chem. 59 1967. PMID: 26824742.
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Keywords: ISAM 140, supplier, ISAM140, high, affinity, adenosine, receptors, A2B, selective, Tocris Bioscience, Adenosine A2B Receptor Antagonist products