Cat. No. 5858
Chemical Name: 1-[1-[4-(4-Fluorophenyl)-4-oxobutyl
Biological ActivityD2 receptor antagonist. Also exhibits affinity for 5-HT, α-adrenergic and histamine receptors,and hERG channels. Antipsychotic and antiemetic.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Rajamani et al (2005) A two-state homology model of the hERG K+ channel: application to ligand binding. Bioorg.Med.Chem.Lett. 15 1737. PMID: 15745831.
Peroutka and Synder (1980) Relationship of neuroleptic drug effects at brain dopamine, serotonin, alpha-adrenergic, and histamine receptors to clinical potency. Am.J.Psychiatry 137 1518. PMID: 6108081.
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Keywords: Droperidol, supplier, dopamine, receptors, D2, antagonists, antipsychotics, antiemetics, herg, channels, Tocris Bioscience, D2 Receptor Antagonist products