JNJ DGAT2-A

Cat. No. 5853

JNJ DGAT2-A C24H16BrFN4O2S

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Chemical Name: 3-Bromo-4-[2-fluoro-4-[[4-oxo-2-[[2-(pyridin-2-yl)ethyl]amino]-1,3-thiazol-5-(4H)ylidene]methyl]phenoxy]benzonitrile

Biological Activity

DGAT2 inhibitor (IC50 = 140 nM). Exhibits >70-fold selectivity for DGAT2 over DGAT1 and MGAT2.

Technical Data

M.Wt:
523.38
Formula:
C24H16BrFN4O2S
Solubility:
Soluble to 100 mM in DMSO
Storage:
Store at +4°C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Product Datasheet / Safety Data Sheet

Qi et al (2012) The use of stable isotope-labeled glycerol and oleic acid to differentiate the hepatic functions of DGAT1 and -2 J.Lipid Res. 53 1106. PMID: 22493088.

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Keywords: JNJ DGAT2-A, supplier, JNJDGAT2-A, Diacylglycerol, O-Acyltransferases, DGAT2, inhibitors, inhibits, Tocris Bioscience, Diacylglycerol O-Acyltransferase Inhibitor products

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