Cat. No. 5837
Biological ActivityHigh affinity rat GIP receptor partial agonist (Kd = 13 nM). Increases cAMP accumulation in COS-7 cells transfected with rat GIP receptor, while also acting as a competitive antagonist of GIP.
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All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Sparre-Ulrich et al (2016) Species-specific action of (Pro3)GIP - a full agonist at human GIP receptors, but a partial agonist and competitive antagonist at rat and mouse GIP receptors. Br.J.Pharmacol. 173 27. PMID: 26359804.
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Keywords: [Pro3]-GIP (Rat), supplier, GIP, receptors, antagonists, antagonism, glucose-dependent, insulinotropic, polypeptide, partial, agonist, agonism, insulin, Tocris Bioscience, GIP Receptor Agonist products