Cat. No. 5762
Chemical Name: N-[(1R)-1-[3-(Cyclopropyloxy)-4-flu
Biological ActivityPotent cholesteryl ester transfer protein (CETP) inhibitor (IC50 = 4 nM in an enzyme-based scintillation proximity assay). Inhibits cholesteryl ester transfer and increases HDL-C levels in vivo. Orally bioavailable.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Qiao et al (2015) Triphenylethanamine derivatives as cholesteryl ester transfer protein inhibitors: discovery of N-[(1R)-1-(3-cyclopropoxy-4-fluorophenyl)-1-[3-fluoro-5-(1,1,2,2-tetrafluoroethoxy)phenyl]-2-phenylethyl]-4-fluoro-3-(trifluoromethyl)benzamide (BMS-795311). J.Med.Chem. 58 9010. PMID: 26524347 .
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Keywords: BMS 795311, supplier, BMS795311, cholesteryl, ester, transfer, protein, CETP, potent, inhibitors, inhibits, orally, bioavailable, high, density, lipoprotein, cholesterol, HDL-C, Tocris Bioscience, Other Transferase Inhibitor products
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