Cat. No. 5761
Alternative Name: RSL1
Chemical Name: 2-Ethyl-3-methoxybenzoic acid 2-(3,5-dimethylbenzoyl)-2-(1,1-dime
Biological ActivityGene switch ligand. Transcription inducer for use in induceable gene expression systems. Does not cause significant changes in endogenous gene expression in HEK cells.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Lapenna et al (2009) Semi-synthetic ecdysteroids as gene-switch actuators: synthesis, structure-activity relationships, and prospective ADME properties. ChemMedChem 4 55. PMID: 19065574.
Panguluri et al (2007) Effect of ecdysone receptor gene switch ligands on endogenous gene expression in 293 cells. FEBS Journal 274 5669. PMID: 17922837.
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Keywords: RG 102240, supplier, RG102240, RheoSwitch, Ligands, inducible, expression, sytems, gene, switch, transcription, ecdysone, receptors, EcR, Tocris Bioscience, Other Transcription Factor products
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